Using chemical fragment binding maps
to discover new possibilities
for optimization of drug compounds
Unique Information: Protein "Hot spots", Chemical Fragment Maps, Water Maps
Easy Energies: Protein-ligand Interactions, Desolvation, Stress
Helpful Services: Docking, Synthesis (Reaxys), Data Mgmt (CDD Vault)

This site is still under development.
Consider any use as experimental.

New proteins: BRD4, BRD9, Bcl-xL, BRPF1, beta catenin with XTCF3-CBD, LXR, NEDD4, FABH.
PDB structures: Download PDB structures for docking, energy calculations on compounds.
Request: Fragment simulations on your favorite PDB structures (click on Contact)!

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Hot Spots Example
Fragment Grow Example